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A new synthetic approach to benzo[4u2019,5u2019]imidazo[2u2019,1u2019:6,1]pyrido[2,3-d]pyrimidine was developed using 2,4,6-trisubstituted pyrimidinyl-5-propanoic acids, overcoming limitations of previous benzimidazole-based methods. This strategy enables functional modifications and enhances biological research potential.
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