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Adrenergic alpha2B Adrenergic alpha2C Adrenergic alpha2: Non-Selective Adrenergic beta1

Acetylcholinesterase Peptidase: Cathepsin G Peptidase Matrix Metalloproteinase-1 Cyclooxygenase COX-1 Cyclooxygenase COX-2 Lipoxygenase 5-LO Monoamine Oxidase MAO-A Monoamine Oxidase MAO-B Nitric Oxide Synthase: Neuronal Nitric Oxide Synthase: Inducible Phosphodiesterase PDE1

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Adrenergic alpha2B Adrenergic alpha2C Adrenergic alpha2: Non-Selective Adrenergic beta1

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  1. Acetylcholinesterase Peptidase: Cathepsin G Peptidase Matrix Metalloproteinase-1 Cyclooxygenase COX-1 Cyclooxygenase COX-2 Lipoxygenase 5-LO Monoamine Oxidase MAO-A Monoamine Oxidase MAO-B Nitric Oxide Synthase: Neuronal Nitric Oxide Synthase: Inducible Phosphodiesterase PDE1 Phosphodiesterase PDE2 Phosphodiesterase PDE3 Phosphodiesterase PDE4 Phosphodiesterase PDE5 Phosphodiesterase PDE6 Peptidase: Caspase 1 Peptidase: Caspase 3 Peptidase: Caspase 6 Peptidase: Caspase 7 Peptidase: Caspase 8 Peptidase: Metalloproteinase: Neutral Endopeptidase Peptidase: Leukocyte Elastase Protein Tyrosine Kinase: EGF Receptor Protein Serine/Threonine Kinase: ERK1 Protein Tyrosine Kinase: Insulin Receptor Protein Serine/Threonine Kinase: p38alpha Protein Tyrosine Kinase: pp60src Protein Serine/Threonine Kinase: PKA: Non-Selective Protein Serine/Threonine Kinase: PKC: Non-Selective Protein Serine/Threonine Kinase: PKCalpha Protein Tyrosine Phosphatase: CD45 Protein Tyrosine Phosphatase: PTP1B Protein Tyrosine Phosphatase: T-Cell Tyrosine Hydroxylase Adenosine A1 Adenosine A2A Adenosine A3 Transporter: Adenosine Adrenergic alpha1D Adrenergic alpha1: Non-Selective Adrenergic alpha2A Adrenergic alpha2B Adrenergic alpha2C Adrenergic alpha2: Non-Selective Adrenergic beta1 Adrenergic beta2 Adrenergic beta3 Transporter: Norepinephrine Angiotensin AT1 Angiotensin AT2 Atrial Natriuretic Factor Bombesin: Non-Selective Bradykinin B2 Calcitonin Calcitonin Gene-Related Peptide CGRP1 Calcium Channel L-Type: Benzothiazepine Calcium Channel L-Type: Dihydropyridine Calcium Channel L-Type: Phenylalkylamine Calcium Channel N-Type Cannabinoid CB1 Cannabinoid CB2 Chemokine CCR1 Chemokine CCR5 Cholecystokinin CCK1 (CCKA) Cholecystokinin CCK2 (CCKB) Transporter: Choline Dopamine D1 Dopamine D2S Dopamine D3 Dopamine D4.4 Dopamine D5 Transporter: Dopamine Endothelin ETA Endothelin ETB Epidermal Growth Factor Estrogen ERalpha Estrogen ERbeta Transporter: GABA GABAA: Agonist Site GABAA: Chloride Channel GABAB: Non-Selective Galanin GAL1 Galanin GAL2 Glucocorticoid Glutamate: AMPA Glutamate: Kainate Glutamate: NMDA: Agonism Glutamate: NMDA: Glycine Glutamate: NMDA: Phencyclidine Glutamate: Non-Selective Glycine: Strychnine-Sensitive Histamine H1 Histamine H2 Histamine H3 Inositol Trisphosphate IP3 Insulin Chemokine CXCR2 (IL-8B) Leukotriene LTD4 Melanocortin MC3 Melanocortin MC4 Melanocortin MC5 Melatonin ML: Non-Selective Transporter: Monoamine Muscarinic M1 Muscarinic M2 Muscarinic M3 Muscarinic M4 Muscarinic M5 Tachykinin NK1 Tachykinin NK2 Tachykinin NK3 Neuropeptide Y1 Neuropeptide Y2 Nicotinic Acetylcholine Opiate delta (OP1: DOP) Opiate kappa (OP2: KOP) Opiate mu (OP3: MOP) Orphanin ORL1 Platelet Activating Factor Potassium Channel [KA] Potassium Channel [KATP] Potassium Channel [SKCA] Purinergic P2X Serotonin 5-HT1: Non-Selective Serotonin 5-HT1A Serotonin 5-HT1B Serotonin 5-HT2: Non-Selective Serotonin 5-HT2A Serotonin 5-HT2B Serotonin 5-HT2C Serotonin 5-HT3 Serotonin 5-HT4 Serotonin 5-HT6 Serotonin 5-HT7 Transporter: Serotonin Sodium Channel: Site 2 Somatostatin sst5 Testosterone Prostanoid: Thromboxane A2 Thyrotropin Releasing Hormone Vasoactive Intestinal Peptide VIP1 Vasopressin V1A Prostanoid EP1 Prostanoid EP3 Prostanoid EP4 Prostanoid FP Prostanoid DP Prostanoid IP Somatostatin sst1 Somatostatin sst2 Somatostatin sst3 Somatostatin sst4 GABA-alpha1beta3gamma2 GABA-alpha1beta3gamma2 GABA-alpha5beta3gamma2 GABA-alpha5beta3gamma2 NMDA-NR1a/NR2a - Antagonist Oxytocin PPAR alpha - Antagonist PPARgamma - Antagonist Bradykinin B1 - Antagonist Neurotensin NT1 - Antagonist Potassium Channel: HERG - Antagonist Vasopressin V1b - Antagonist Vasopressin V2 - Antagonist Supplemental TABLE List of the 166 target molecules screened at MDS Pharma

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