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Peptide receptors

Non-peptide receptors. Peptide receptors. Adenosine. A1 (h). Angiotensin-II. AT1 (h). A2A (h). AT2 (h). Bombesin. bb3 (h). A2B (h). B2 (h). A3 (h). Calcitonin gene-related peptide. CGRP (h). Adrenergic. alpha 1A (h). Chemokine. CCR1 (h). alpha 2A (h). Cholecystokinin. CCKA (h).

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Peptide receptors

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  1. Non-peptide receptors Peptide receptors Adenosine A1 (h) Angiotensin-II AT1 (h) A2A (h) AT2 (h) Bombesin bb3 (h) A2B (h) B2 (h) A3 (h) Calcitonin gene-related peptide CGRP (h) Adrenergic alpha 1A (h) Chemokine CCR1 (h) alpha 2A (h) Cholecystokinin CCKA (h) alpha 2B (h) CCKB (h) alpha 2C (h) Complement 5a C5a (h) beta 1 (h) Endothelin ETA (h) beta 2 (h) ETB (h) beta 3 (h) Galanin GAL1 (h) Cannabinoid CB1 (h) Glucagon Glucagon (h) CB2 (h) Growth hormone secretagogue Ghrelin (h) Dopamine D1 (h) Melanin-concentrating hormone MCH1 (h) D2S (h) MC1 (m) D3 (h) MC3 (h) D4.4 (h) MC4 (h) GABA GABAA (r) Motilin Motilin (h) GABAB(1b) (h) Neurokinin NK1 (h) BZD (central) (r) NK2 (h) Cl- channel (r) Neuropeptide Y Y1 (h) Glutamate AMPA (r) Neurotensin NT1 (h) Kainate (r) Opioid and opioid-like delta 2 (h) NMDA (r) kappa (h) PCP (r) mu (h) Glycine (strychnine-insensitive) (r) Glycine ORL1 (h) Glycine (strychnine-sensitive) (r) Somatostatin sst4 (h) Histamine H1 (h) sst5 (h) H2 (h) Thyroid hormone TH (r) Urotensin-II UT1 (h) H3 (h) Vasoactive intestinal peptide VIP1 (h) Imidazole I1(b) PACAP (h) Leukotriene LTD4 (h) Vasopressin V1a (h) Melatonin ML1 (c) V1b (h) ML2 (MT3) (ham) V2 (h) Muscarinic M1 (h) Ion channels M2 (h) Ca2+ channels Ca2+ channel (L, DHP site) M3 (h) Ca2+ channel (L, diltiazem site) M4 (h) M5 (h) Ca2+ channel (L, verapamil site) Nicotinic N (neuronal) (α-BGTX-insensitive) (r) Ca2+ channel (N) N (muscle-type) (h) Ryanodine (RY3) Purinergic P2X (r) Serotonin 5-HT1A (h) K+ channels K+ATP channel (r) 5-HT1B (h) K+V channel (r) 5-HT1D (r) SK+Ca channel (r) 5-HT2A (h) Na+ channel Na+ channel (site 2) 5-HT2B (h) (agonist site) 5-HT2C (h) 5-HT3 (h) Amine transporter 5-HT4e (h) Choline NE transporter (h) 5-HT6 (h) Dopamine DA transporter (h) 5-HT7 (h) GABA GABA transporter sigma (non-selective) (r) Sigma Norepinephrine Choline transporter (h) 5-HT transporter (h) Seretonin Nuclear receptors Glucocorticoid GR (h) Estrogen alpha Eralpha (h) AR (h) Androgen Enzymes Phosphodiesterases PDE2 (h) PDE3 (h) PDE4 (h) PDE5 (h) PDE6 (b) Arachidonic acid/ COX1 (h) prostaglandin metabolism COX2 (h) PGE2 secretion (h) Monoamine and neurotransmitter MAO-A (h) synthesis and metabolism MAO-B (h) GABA transaminase (r) Acetylcholinesterase (h) COMT (Catechol- O-methyl transferase) (p) Histamine N-Methyltransferase (h) Tyrosine hydroxylase (r) Nitric oxide synthesis Cerebellar constitutive NOS (r) Endothelial constitutive NOS (h) Second messenger systems Guanylyl cyclase (b) ATPases ATPase (Na+/K+) (d) Lipid synthesis HMG-CoA reductase (ham) Miscellaneous enzymes Carbonic anhydrase II (h) Xanthine oxidase Kinases Phosphatases Phospholipases Proteases CaMK2α (h) ERK2 (h) p56Fyn kinase (h) p55Lyn kinase (h) ZAP70 kinase (h) Abl kinase (h) Protein kinase C (r) Protein kinase B-α (h) CDK1 Phosphatase 1B (h) Phosphatase C (r) Elastase (h) Tryptase (h) ACE (h) BACE-1 (h) TACE (h) HIV-1 protease (h) ACE (h) Neutral endopeptidase (h) MMP-1 (h) MMP-2 (h) MMP-3 (h) MMP-7 (h) MMP-9 (h) Cathepsin X (h) Cathepsin L (h) Cathepsin H (h) Cathepsin G (h) Cathepsin E (h) Cathepsin D (h) Cathepsin B (h) m-Calpain (r) m-Calpain (h) Granzyme B (h) Supplementary Table 3, Chauvier et al..2011

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